Is Sublingual Administration Safe for Nootropics?

nootropics sublingual

Nootropics can boost your creativity.

Sublingual administration is one of many ways to take a supplement for maximum effect.  It is done by putting a supplement under the tongue and allowing it to diffuse into the bloodstream through the mucous membrane beneath the tongue.  Taking substances this way can lead to faster effects because they go straight into the bloodstream rather than being passed through the liver first or being degraded by stomach acid.

While this seems like an effective way to take nootropic supplements, many users may wonder if this method is safe.  While the majority of nootropics are perfect safe to take sublingually, some are better than others to ingest this way.

Which Supplements Can I Take Sublingually?

The effects of taking a nootropic sublingually depend on the composition of the substance.  Anything that is more acidic, like phenibut, may make the mouth sore, as do substances like adrafinil.  Some are just not as effective because they dissolve slowly, like sulbutiamine.

nootropics writing

Nootropics can also boost your writing ability.

These types of supplements are best taken orally with water or juice for optimal safety and efficacy.  The ideal nootropic for sublingual administration is one that dissolves quickly and is more effective when it is absorbed directly into the bloodstream and skips the liver.

Racetam supplements, like aniracetam and coluracetam, as well as derivatives like noopept, are much more effective when they are absorbed into the tongue’s mucous membrane.  Nootropics like Alpha GPC also dissolve quickly, and have no associated taste. It also helps that many nootropics, coluracetam and noopept in particular, have very minute dosages which makes sublingual supplementation much easier.

Is It Better To Take Nootropics Sublingually?

sublingual nootropics

Sublingual administration involves putting the supplement under your tongue.

Sublingual administration is not necessarily better or worse than oral administration, and choosing to take nootropics this way entirely depends on the needs of the individual.  Taking nootropics beneath the tongue allows the user to take smaller doses because they are more effective, more concentrated, and work faster.

Also, users trying to avoid stress on the stomach and intestinal tract may take supplements sublingually to avoid side effects related to the digestive system.  Bypassing the stomach also means better absorption and less degradation, making the supplement more potent [1].

While sublingual administration seems better and more effective, it can be difficult to find nootropics designed to be taken this way. Generally, racetams as well as l-theanine and vitamin B6 will be widely available this way.  Otherwise, many supplements are only intended for oral administration.

The Safest Way to Take Nootropics with Sublingual Administration

The best way to remain safe when taking nootropics is to follow the instructions and dosages and only use sublingual administration when the supplement is intended for this form of absorption.  These supplements are entirely safe when taken as intended, but may irritate the mouth if used incorrectly.

As with any supplement, it’s best to pay attention to the guidelines to enjoy maximum positive effects.  However, finding nootropics designed to be taken sublingually can be a great way to enjoy quick and powerful cognitive effects without losing significant amounts of the supplement as the body breaks it down.



ALCAR Benefits

Choline is an essential nutrient that serves as both a nootropic supplement and an athletic performance enhancer. Choline supplements cause the release of acetylcholine, which improves memory and mood as well as allowing better communication between nerve cells and muscle cells.

Since choline has multiple benefits, it makes sense to use as a dietary supplement.  However, using choline on a regular basis or several times a day can cause some people to experience the “choline blues.”

This refers to a slight depressive state that can be stopped by discontinuing use of the supplement for a period of time.  Rather than dealing with the blues, individuals can take an alternative supplement, ALCAR, to experience the same effects.

ALCAR versus Choline

ALCAR, also known as Acetyl-L-carnitine, is a modified amino acid that has a variety of health benefits.  Like Choline, it causes increased production of acetylcholine, as well as dopamine, the feel-good hormone.

Its main function is helping the body to break down fatty acids and produce energy, but it also works as a neuroprotectant, removing damaged fats from the brain and strengthening neural connections.

While Choline can delay fatigue for athletes, ALCAR can actually help with muscle recovery [1].  ALCAR helps to regulate carnitine levels, which are essential for the conversion of fat to energy, while supplemental choline mostly gives an extra boost at the end of a workout or athletic event.

Though they both increase acetylcholine, ALCAR has a few more benefits and doesn’t result in any negative mood reactions.

ALCAR Benefits Continued

A very important benefit of ALCAR is its ability to break down fats, both for energy production and to rid the brain of harmful fatty acids.

It can easily cross the blood-brain barrier, which is why is has such powerful mental effects.  While the supplement can increase alertness and elevate mood, it also protects to brain against deterioration and keeps the nervous system healthy.

Additionally, this supplement can lower blood pressure to improve heart health, reduce anxiety and feelings of stress, and even increase fertility in men.  Most significantly, ALCAR doesn’t produce anything similar to “choline blues” since it boosts dopamine.

ALCAR Benefits Vs Choline

ALCAR is entirely safe in dosages between 300 and 500 milligrams, and shouldn’t produce any noticeable side effects if taken correctly.  It’s natural, has a wide array of benefits, and is perfect for both athletes and nootropic users.

Anyone experiencing the blues while taking choline supplementsshould consider trying ALCAR as an easy way to feel better both physically and mentally.