Is Sublingual Administration Safe for Nootropics?

nootropics sublingual

Nootropics can boost your creativity.

Sublingual administration is one of many ways to take a supplement for maximum effect.  It is done by putting a supplement under the tongue and allowing it to diffuse into the bloodstream through the mucous membrane beneath the tongue.  Taking substances this way can lead to faster effects because they go straight into the bloodstream rather than being passed through the liver first or being degraded by stomach acid.

While this seems like an effective way to take nootropic supplements, many users may wonder if this method is safe.  While the majority of nootropics are perfect safe to take sublingually, some are better than others to ingest this way.

Which Supplements Can I Take Sublingually?

The effects of taking a nootropic sublingually depend on the composition of the substance.  Anything that is more acidic, like phenibut, may make the mouth sore, as do substances like adrafinil.  Some are just not as effective because they dissolve slowly, like sulbutiamine.

nootropics writing

Nootropics can also boost your writing ability.

These types of supplements are best taken orally with water or juice for optimal safety and efficacy.  The ideal nootropic for sublingual administration is one that dissolves quickly and is more effective when it is absorbed directly into the bloodstream and skips the liver.

Racetam supplements, like aniracetam and coluracetam, as well as derivatives like noopept, are much more effective when they are absorbed into the tongue’s mucous membrane.  Nootropics like Alpha GPC also dissolve quickly, and have no associated taste. It also helps that many nootropics, coluracetam and noopept in particular, have very minute dosages which makes sublingual supplementation much easier.

Is It Better To Take Nootropics Sublingually?

sublingual nootropics

Sublingual administration involves putting the supplement under your tongue.

Sublingual administration is not necessarily better or worse than oral administration, and choosing to take nootropics this way entirely depends on the needs of the individual.  Taking nootropics beneath the tongue allows the user to take smaller doses because they are more effective, more concentrated, and work faster.

Also, users trying to avoid stress on the stomach and intestinal tract may take supplements sublingually to avoid side effects related to the digestive system.  Bypassing the stomach also means better absorption and less degradation, making the supplement more potent [1].

While sublingual administration seems better and more effective, it can be difficult to find nootropics designed to be taken this way. Generally, racetams as well as l-theanine and vitamin B6 will be widely available this way.  Otherwise, many supplements are only intended for oral administration.

The Safest Way to Take Nootropics with Sublingual Administration

The best way to remain safe when taking nootropics is to follow the instructions and dosages and only use sublingual administration when the supplement is intended for this form of absorption.  These supplements are entirely safe when taken as intended, but may irritate the mouth if used incorrectly.

As with any supplement, it’s best to pay attention to the guidelines to enjoy maximum positive effects.  However, finding nootropics designed to be taken sublingually can be a great way to enjoy quick and powerful cognitive effects without losing significant amounts of the supplement as the body breaks it down.

Sources

1. http://www.examiner.com/article/new-methods-of-nootropic-administration

ALCAR Benefits

Choline is an essential nutrient that serves as both a nootropic supplement and an athletic performance enhancer. Choline supplements cause the release of acetylcholine, which improves memory and mood as well as allowing better communication between nerve cells and muscle cells.

Since choline has multiple benefits, it makes sense to use as a dietary supplement.  However, using choline on a regular basis or several times a day can cause some people to experience the “choline blues.”

This refers to a slight depressive state that can be stopped by discontinuing use of the supplement for a period of time.  Rather than dealing with the blues, individuals can take an alternative supplement, ALCAR, to experience the same effects.

ALCAR versus Choline

ALCAR, also known as Acetyl-L-carnitine, is a modified amino acid that has a variety of health benefits.  Like Choline, it causes increased production of acetylcholine, as well as dopamine, the feel-good hormone.

Its main function is helping the body to break down fatty acids and produce energy, but it also works as a neuroprotectant, removing damaged fats from the brain and strengthening neural connections.

While Choline can delay fatigue for athletes, ALCAR can actually help with muscle recovery [1].  ALCAR helps to regulate carnitine levels, which are essential for the conversion of fat to energy, while supplemental choline mostly gives an extra boost at the end of a workout or athletic event.

Though they both increase acetylcholine, ALCAR has a few more benefits and doesn’t result in any negative mood reactions.

ALCAR Benefits Continued

A very important benefit of ALCAR is its ability to break down fats, both for energy production and to rid the brain of harmful fatty acids.

It can easily cross the blood-brain barrier, which is why is has such powerful mental effects.  While the supplement can increase alertness and elevate mood, it also protects to brain against deterioration and keeps the nervous system healthy.

Additionally, this supplement can lower blood pressure to improve heart health, reduce anxiety and feelings of stress, and even increase fertility in men.  Most significantly, ALCAR doesn’t produce anything similar to “choline blues” since it boosts dopamine.

ALCAR Benefits Vs Choline

ALCAR is entirely safe in dosages between 300 and 500 milligrams, and shouldn’t produce any noticeable side effects if taken correctly.  It’s natural, has a wide array of benefits, and is perfect for both athletes and nootropic users.

Anyone experiencing the blues while taking choline supplementsshould consider trying ALCAR as an easy way to feel better both physically and mentally.

Sources

1. http://www.ncbi.nlm.nih.gov/pubmed/1864226

Piracetam, Noopept, Theanine and Caffeine: Hack your Brain for Increased Productivity

You’re going to run a marathon. You’ve already decided. Well, in your heart at least, because you still haven’t gotten off the couch to start that elaborate training routine you’ve come up with.

So what do you do in the meantime? Dream up how great it will be when you finally run. The adrenaline as you pass over the finish line, the cheers from your friend and family, the pride that you’ll feel. Dreaming big will make sure that you act big, won’t it? After all, you need concrete goals to get anywhere.

Take those big dreams, toss in some supplements for focus, maybe a few more supplements for concentration, and you’re pretty much guaranteed to succeed. Right?

Unfortunately some recent studies indicate not necessarily [1]. One study had some participants envision a happy resolution to a crisis in another country, while the rest were just asked to state the facts of the crisis. When later asked to donate $25 or more, it turns out the participants who only recited cold facts were much more likely to donate.

The results were repeated in two more trials. One used similar procedures (this time related to donating time to a charity) while the other replaced stating the facts with imagining wasting time — establishing that it wasn’t stating facts that increased will to act, but it was positive dreaming that reduced it.

The takeaway here is that, to a certain extent, positive fantasies reduce the amount of effort you’re willing to put into making that fantasy come true. The downside is that it’s not exactly easy to quit daydreaming. Every second you spend distracted from a task is very likely a second you’re going to spend imagining how great it will feel once you finish.

Fortunately with nootropics, it’s not just a matter of you trying to force yourself to focus. By adding a few crucial supplements for focus to your daily routine, you can watch your concentration skyrocket. Less time dreaming, more time doing — what more could you ask for?

Piracetam

Start off your pursuit of boosted concentration with piracetam powder, one of the oldest and most widely researched nootropics out there. Before we go any further on its concentration-boosting benefits, take a moment to consider that piracetam also shows promise for positive effects on cognition, learning, and memory [1]. If your area-of-needed focus is academic or otherwise cognitively oriented, you’re looking at added benefits from piracetam straight from the get go.

On to its benefits for focus and concentration: Piracetam has repeatedly shown itself to benefit both, allowing users to participate in tasks for longer, less interrupted stints — it makes cognitive flow easier. Piracetam, an AMPA modulator, induces this effect by increasing the amount of oxygen that gets to the brain [2]. Communication between brain hemispheres is boosted, manifesting as a feeling of focus and clarity.

Noopept

If piracetam isn’t quite cutting it or you’re just looking to up your edge even further, check out noopept. It’s actually derived from the racetam family, meaning that it has some similarities to piracetam. It’s definitely its own beast though, and you’ll find a clear cut illustration of the differences before you even start to read up on the effects. While a typical piracetam dose will run between 1 to 3 grams, noopept powder is about a thousand times stronger, working efficiently at doses as small as 10 mg [3].

This might make you think it’s simply a jacked up piracetam, but noopept has its own distinct effects. Noopept is touted for anti-anxiety benefits in addition to its cognitive gains [4]. The upshot of this is that you spend less time worrying — if you aren’t worrying, it’s a heck of a lot easier to stop working. Add in the facts that noopept has shown to be neuroprotective and that its effects actually build over time [5], and you’re looking at a very potent productivity aid.

Caffeine and Theanine

Last but not least, a knock-out combo that will see your morning coffee benefiting you in completely new ways. While both of the following are effective supplements for concentration on their own, mixing l-theanine and caffeine powder will produce a synergistic effect that goes well beyond what you’d get from taking either individually.

Theanine is actually an amino acid that you’ve probably come across before without realizing it: it’s found in green tea. Taken on its own, it affects both your GABA and glutumate receptors, and is well-documented for having calming, relaxing effects [6].

Caffeine on its own stimulates a whole slew of neurotransmitters, but leaves you feeling wired and sets you up for an eventual crash. Together? Theanine takes the edge off of caffeine, smooths out the comedown, and makes it much easier to focus. A trialed study found that participants on a combination of theanine and caffeine were much better at focusing on difficult cognitive tasks [7]. So next time you grab a coffee to give yourself energy boosts, add in some theanine – and unlock your full potential.

Focus and concentration don’t come easy, and even with nootropic supplementation require discipline and practice. With the right stack, though, it’s possible to “hack” your brain into increased productivity. Experiment with combinations and compounds, find what works best for you, and boot those endless daydreams out of your head!

Sources

  1. http://www.psychologytoday.com/blog/ulterior-motives/201302/positive-fantasies-can-reduce-future-effort
  2. http://examine.com/supplements/Piracetam/
  3. http://www.ncbi.nlm.nih.gov/pubmed/12596521
  4. http://examine.com/supplements/Noopept/
  5. http://www.braintropic.com/noopept/
  6. http://examine.com/supplements/Theanine/
  7. http://www.ncbi.nlm.nih.gov/pubmed/18681988